Synthesis and receptor binding of new thieno[2,3-d]pyrimidines as selective ligands of 5-HT3 receptors
With the aim to develop new potent and selective ligands of 5-HT3-type serotonin receptors and to acquire more information on their structure-affinity relationships, new thieno[2,3-d]pyrimidine derivatives 32-39 were synthesized and their binding to 5-HT3 versus 5-HT4 receptors was studied. Some of...
Elmentve itt :
Szerzők: |
Modica Maria N. Romeo Giuseppe Salerno Loredana Pittala Valeria Siracusa Maria A. Mereghetti Ilario Cagnotto Alfredo Mennini Tiziana Gáspár Róbert Gál Adrienn Falkay György Palkó Márta Maksay Gábor Fülöp Ferenc |
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Dokumentumtípus: | Cikk |
Megjelent: |
2008
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Sorozat: | ARCHIV DER PHARMAZIE
341 No. 6 |
doi: | 10.1002/ardp.200700205 |
mtmt: | 1127905 |
Online Access: | http://publicatio.bibl.u-szeged.hu/16155 |
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